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result sql = Synthesis and structure-activity relationships of oxime neurokinin antagonists: discovery of potent arylamides.
Synthesis and structure-activity relationships of oxime neurokinin antagonists: discovery of potent arylamides.
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result sql = The structural modification of the benzylic ether region of oxime 1 has resulted in the identification of several novel aryl amides as selective or dual NK(1)/NK(2) antagonists.

Publication: Bioorg. Med. Chem. Lett. 2002 Jan 21 ;12(2)::141-5.
Publication Date: 2002 Jan 21
Study Author(s): Shih, Neng Yang;Albanese, Margaret;Anthes, John C;Carruthers, Nicholas I;Grice, Cheryl A;Lin, Ling;Mangiaracina, Pietro;Reichard, Gregory A;Schwerdt, John;Seidl, Vera;Wong, Shing-Chung;Piwinski, John J;
Institution: Schering-Plough Research Institute, 2015 Galloping Hill Rd, Kenilworth, NJ 07033-1300, USA. [email protected]
Shortcut link to this study:
The structural modification of the benzylic ether region of oxime 1 has resulted in the identification of several novel aryl amides as selective or dual NK(1)/NK(2) antagonists.
PMID: 11755340

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