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result sql = Enhanced anti-tumor effect of combination therapy with gemcitabine and apigenin in pancreatic cancer.
Enhanced anti-tumor effect of combination therapy with gemcitabine and apigenin in pancreatic cancer.
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result sql = Apigenin is a dietary flavonoid possessing therapeutic potential against cancers. This study was designed to investigate whether combination therapy with gemcitabine and apigenin enhanced anti-tumor efficacy in pancreatic cancer. In vitro, the combination treatment resulted in more growth inhibition and apoptosis through the down-regulation of NF-kappa B activity with suppression of Akt activation in pancreatic cancer cell lines (MiaPaca-2, AsPC-1). In vivo, the combination therapy augmented tumor growth inhibition through the down-regulation of NF-kappa B activity with the suppression of Akt in tumor tissue. The combination of gemcitabine and apigenin enhanced anti-tumor efficacy through Akt and NF-kappa B activity suppression and apoptosis induction.

Publication: Cancer Lett. 2008 Jan 18 ;259(1)::39-49.
Publication Date: 2008 Jan 18
Study Author(s): Lee, Sang Hyub;Ryu, Ji Kon;Lee, Kyeung-Yeup;Woo, Sang Myung;Park, Joo Kyung;Yoo, Ji Won;Kim, Yong-Tae;Yoon, Yong Bum;
Institution: Department of Internal Medicine and Liver Research Institute, Seoul National University College of Medicine, 110-744, Yeongeon-dong 28, Jongno-gu, Seoul, Republic of Korea.
Shortcut link to this study:
Apigenin is a dietary flavonoid possessing therapeutic potential against cancers. This study was designed to investigate whether combination therapy with gemcitabine and apigenin enhanced anti-tumor efficacy in pancreatic cancer. In vitro, the combination treatment resulted in more growth inhibition and apoptosis through the down-regulation of NF-kappa B activity with suppression of Akt activation in pancreatic cancer cell lines (MiaPaca-2, AsPC-1). In vivo, the combination therapy augmented tumor growth inhibition through the down-regulation of NF-kappa B activity with the suppression of Akt in tumor tissue. The combination of gemcitabine and apigenin enhanced anti-tumor efficacy through Akt and NF-kappa B activity suppression and apoptosis induction.
PMID: 17967505

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