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result sql = Overcoming the drug resistance in breast cancer cells by rational design of efficient glutathione S-transferase inhibitors.
Overcoming the drug resistance in breast cancer cells by rational design of efficient glutathione S-transferase inhibitors.
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result sql = A new type of competitive human GST inhibitors has been developed via the bioisostere and structure activity profile strategies; we report their discovery, preparation, inhibitory activity, and synergetic effect in combination with chemotherapy drugs against breast cancer cells.

Publication: Org. Lett. 2010 Jan 1 ;12(1)::20-3. :doi: 10.1021/ol902298s.
Publication Date: 2010 Jan 1
Study Author(s): Li, Wen-Shan;Lam, Wing See;Liu, Kung-Cheng;Wang, Chie-Hong;Chang, Hui Chuan;Jen, Ya Ching;Hsu, Yu-Ting;Shivatare, Sachin S;Jao, Shu-Chuan;
Institution: Institute of Chemistry, Academia Sinica, Taipei 115, Taiwan. [email protected]
Shortcut link to this study:
A new type of competitive human GST inhibitors has been developed via the bioisostere and structure activity profile strategies; we report their discovery, preparation, inhibitory activity, and synergetic effect in combination with chemotherapy drugs against breast cancer cells.
PMID: 19961147

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